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GPCR Therapeutics

GPCR Therapeutics

Private
SeoulHealthcare & Life Scienceshttp://gpcr.co.kr/

Last Round

Private Equity

Jul 2, 2026

Est. Valuation

$53.56M

Total Funding Raised

$108.83M

Company Overview

GPCR Therapeutics is a biopharmaceutical company that develops innovative cancer therapeutics by targeting G protein-coupled receptor (GPCR) heteromers.

Sector

Healthcare & Life Sciences

Verticals

Biotechnology, Drug Discovery

Business Model

B2B

Customer Profile

Revenue Share, Services & Consulting

AI Layer

Non-AI

Keywords

GPCRdrug discoverybiotechtherapeutic developmentoncologyrespiratory diseaseantibody therapeuticssmall moleculeout-licensingbiopharmaclinical-stage biotechdrug pipelinemultiple myelomaidiopathic pulmonary fibrosisIPF

Historical Pricing

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GPCR Therapeutics Comps

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GPCR Therapeutics comps — public and private peers by sector, stage, and business model
CompanyStatusEst. ValuationRev Multiple
OpenAIPrivate$86.0B~40x
CoherePrivate$5.0B--
Competitor 1Public$XX.XBXXx
Competitor 2Public$XX.XBXXx

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GPCR Therapeutics Funding Rounds

Historical fundraising activity

Data table
RoundDateAmount RaisedValuationInvestorsSources
Private EquityJul 2, 2026
Series C ExtensionNov 1, 2023
Series CJun 30, 2021
Series CApr 30, 2021
Series BJul 31, 2019
Series A
Sep 30, 2016

GPCR Therapeutics Investors

Notable investors and investment history

GPCR Therapeutics investors
InvestorRounds
InterVestSeries B, Series C, Series A
Kinggo Investment PartnersSeries C Extension
Smilegate InvestmentSeries B, Series C
Kingo Investment PartnersSeries C Extension
SUNP CorporationSeries C
Company K PartnersSeries C, Series A
Medytox Venture InvestmentSeries B, Series C Extension

Market signals

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  • Nov 23, 2023

    $3.15M round led by Medytox Venture Investment

  • Sep 30, 2016

    Raised $9.35M from Company K Partners and InterVest.

GPCR Therapeutics Filings

SEC and related filings with document metadata.

Data table
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GPCR Therapeutics Filings

SEC and related filings with document metadata.

Frequently Asked Questions

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Firmographic Details

HeadquartersSeoul
Employee Range16
Year Founded2013
Last FundingJul 2, 2026

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