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BTB Therapeutics, Inc.

BTB Therapeutics, Inc.

Private
Escondido, CaliforniaHealthcare & Life Scienceshttps://www.btbtherapeutics.com/en/

Last Round

Seed Round

Aug 12, 2026

Est. Valuation

$6.42M

Total Funding Raised

$11.96M

Momentum

Top 5%

of companies Caplight tracks

Company Overview

BTB Therapeutics, Inc. is a drug discovery company developing non-opioid analgesics and RNA-modifying compounds to treat rare genetic diseases and enhance cancer immunotherapy.

Sector

Healthcare & Life Sciences

Verticals

Biotechnology, Drug Discovery, Clinical Trials

Business Model

B2B

Customer Profile

Services & Consulting

AI Layer

Non-AI

Keywords

non-opioid analgesicpain managementdrug discoveryRNA splicingbiotechtranscriptomicsimmuno-oncologyrare diseasesmall moleculeclinical-stagenon-addictive painkillerdrug licensingbiopharmatherapeutic development

Historical Pricing

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Caplight Momentum Score

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BTB Therapeutics, Inc. Comparables

Compare BTB Therapeutics, Inc. with similar companies based on industry and business-model similarity.

BTB Therapeutics, Inc. comparables — related companies by embedding similarity
CompanySimilarityMarket Cap
Neumentum, Inc.
86%
Allay Therapeutics
84%
Concentric Analgesics
83%

BTB Therapeutics, Inc. Funding Rounds

Historical fundraising activity

Data table
RoundDateAmount RaisedValuationInvestorsSources
Seed RoundAug 12, 2026
Early FundingNov 1, 2025
SeedFeb 5, 2025
Convertible DebtJun 24, 2024
Convertible DebtOct 27, 2023
VC Round
Apr 4, 2023

Key People

Founding team and executive leadership

Masatoshi Hagiwara

Founder Chief Scientific Officer

Founding Team

Takashi Kiyoizumi

Chief Executive Officer

Executive Team

BTB Therapeutics, Inc. Investors

Notable investors and investment history

BTB Therapeutics, Inc. investors
InvestorRounds
Kyoto University Innovation CapitalEarly Funding, Convertible Debt, Seed
SMBC Venture CapitalEarly Funding, Convertible Debt

Market signals

Structured signals derived from secondary market and firmographic data.

  • Aug 12, 2026

    Raised $9M in Seed funding.

  • Nov 1, 2025

    $7M raised in early funding.

BTB Therapeutics, Inc. Filings

SEC and related filings with document metadata.

Data table
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BTB Therapeutics, Inc. Filings

SEC and related filings with document metadata.

Frequently Asked Questions

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Firmographic Details

HeadquartersEscondido, California
Employee Range7
Year Founded2020
Last FundingAug 12, 2026

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